Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of kd data for polymerid = 50000354,50001081,50002497
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50389432(CHEMBL2064618)
Affinity DataKd:  1.73nMAssay Description:Binding affinity to VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma counting in presence of haloperidolMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50292902((2R,3R)-3-(4-(aminomethyl)-4-phenylpiperidin-1-yl)...)
Affinity DataKd:  3nMAssay Description:Displacement of [3H]vesamicol from human vesicular acetylcholine transporter expressed in rat PC12 cells by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50009602(2-(4-Phenyl-piperidin-1-yl)-cyclohexanol | CHEMBL8...)
Affinity DataKd:  7.40nMAssay Description:Binding affinity to VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma counting in presence of DTGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Kanazawa University

Curated by ChEMBL
LigandPNGBDBM50389434(CHEMBL2064619)
Affinity DataKd:  17.4nMAssay Description:Binding affinity to VAChT in rat cerebral membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed